Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50006582
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50051165(8-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-8-az...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50051166(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrr...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  8.20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  12.3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50051164(2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-isoi...)
Affinity DataKi:  140nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50051168(8-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethyl]-8-az...)
Affinity DataKi:  1.33E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50051167(1-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-pyrr...)
Affinity DataKi:  2.92E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50051163(2-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethyl]-isoi...)
Affinity DataKi:  4.13E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM13016(1,2,3,4-tetrahydroisoquinoline | THIQ 6 | tetrahyd...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed