Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50006501
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033666({[2-(2-Amino-6-oxo-1,6-dihydro-purin-9-ylmethoxy)-...)
Affinity DataKi:  10nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049967([4-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  48nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049963([7-(6-Amino-4-oxo-4,5-dihydro-pyrazolo[3,4-d]pyrim...)
Affinity DataKi:  49nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049969(Phosphoric acid mono-[4-(2-amino-6-oxo-1,6-dihydro...)
Affinity DataKi:  51nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049966([4-(2-Amino-6-oxo-1,6-dihydro-purin-9-ylmethoxy)-b...)
Affinity DataKi:  56nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049971([7-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-1,1-difl...)
Affinity DataKi:  57nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049954([5-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  65nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049959([5-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  96nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049972([5-(2-Amino-6-oxo-1,6-dihydro-purin-9-ylmethoxy)-p...)
Affinity DataKi:  160nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049957([6-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  190nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049968([6-(2-Amino-6-oxo-1,6-dihydro-purin-9-ylmethoxy)-h...)
Affinity DataKi:  220nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049955([5-(6-Amino-4-oxo-4,5-dihydro-pyrazolo[3,4-d]pyrim...)
Affinity DataKi:  230nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049960([6-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  360nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049961([8-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-octyl]-p...)
Affinity DataKi:  390nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049962([7-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-heptyl]-...)
Affinity DataKi:  530nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049958([5-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  550nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049970([7-(6-Amino-4-oxo-4,5-dihydro-pyrazolo[3,4-d]pyrim...)
Affinity DataKi:  580nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049964([6-(6-Amino-4-oxo-4,5-dihydro-pyrazolo[3,4-d]pyrim...)
Affinity DataKi:  630nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049956([8-(6-Amino-4-oxo-4,5-dihydro-pyrazolo[3,4-d]pyrim...)
Affinity DataKi:  1.10E+3nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049965([10-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-decyl]-...)
Affinity DataKi:  1.60E+3nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50049973([4-(5-Amino-7-oxo-6,7-dihydro-[1,2,3]triazolo[4,5-...)
Affinity DataKi:  7.30E+3nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase isolated from human erythrocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed