Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50036485
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049199(L-159894 | 4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041969(3-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030711(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030711(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049181(2-Butyl-3-(2'-(butyloxycarbonylaminosulphonyl)-bip...)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032353(isopentyloxy 2-[2-(4-{4-ethyl-5-[3-[3-pyridyl(prop...)
Affinity DataIC50: 0.280nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049203(N-[7-Methyl-2-propyl-3-(2'-isopentyloxycarbonylsul...)
Affinity DataIC50: 0.290nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049214(2-Ethyl-5,7-dimethyl-3-[5'-propyl-2'-(1H-tetrazol-...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50031491(3-(2'-Propylaminocarbonylsulfamoyl-biphenyl-4-ylme...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50009718(CHEMBL7550 | 2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetraz...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049185(L-162620 | Imidazo[4,5-b]pyridine derivative | 4'-...)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049204(L-163579 | 4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ure...)
Affinity DataIC50: 0.390nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035451(4'-[3-Butyl-5-oxo-1-(2-trifluoromet hyl-phenyl)-15...)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049204(L-163579 | 4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ure...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049198(3-{2-Butyl-7-methyl-3-[2'-(2H-tetrazol-5-yl)-biphe...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049182(PD-126055 | (S)-5-Benzyloxy-2-diphenylacetyl-6-met...)
Affinity DataIC50: 0.600nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049206(Biphenylsulfonylcarbamate compound | 5-Ethyl-3-(3-...)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM82433(L-159689 | CHEMBL302102 | N-Pentyl-N-[[2-propyl-3-...)
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049185(L-162620 | Imidazo[4,5-b]pyridine derivative | 4'-...)
Affinity DataIC50: 0.940nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049189(butyl 3-(4-((2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369183(L-163491 | CHEMBL290214)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049195(L-162389 | 3-[(2'-(butylsulfonylcarbamate)-3'-prop...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049183(2,7-Diethyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity was evaluated against angiotensin II type 1 rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM82433(L-159689 | CHEMBL302102 | N-Pentyl-N-[[2-propyl-3-...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049179(L-161570 | 4'-(4-Ethyl-5-formyl-2-propyl-imidazol-...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049189(butyl 3-(4-((2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049214(2-Ethyl-5,7-dimethyl-3-[5'-propyl-2'-(1H-tetrazol-...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049181(2-Butyl-3-(2'-(butyloxycarbonylaminosulphonyl)-bip...)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50041963({2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Guinea pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049187(ZD-7155 | 5,7-Diethyl-1-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 3.80nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in guinea pig adrenal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049193(9,28-dipropyl-13-sulfurdioxo-1,14,22,27-tetraazape...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049178(2-Propyl-5-(4-pyridin-2-yl-piperazin-1-ylmethyl)-3...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Guinea pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50047126(2-Ethyl-4-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 5nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in guinea pig adrenal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049197([5-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043469({Allyl-[4-(2-ethyl-5,7-dimethyl-imidazo[4,5-b]pyri...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049195(L-162389 | 3-[(2'-(butylsulfonylcarbamate)-3'-prop...)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049200(2-Ethyl-5,7-dimethyl-3-[9-(1H-tetrazol-5-ylmethyl)...)
Affinity DataIC50: 11nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in rat adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049202(CGP-42112A | (2S,3R)-2-({(S)-1-[(S)-2-[(S)-2-[(S)-...)
Affinity DataIC50: 12nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049180(L-162132 | (S)-1-Diphenylcarbamoyl-4-{pentyl-[2'-(...)
Affinity DataIC50: 15nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50035451(4'-[3-Butyl-5-oxo-1-(2-trifluoromet hyl-phenyl)-15...)
Affinity DataIC50: 17nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049199(L-159894 | 4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50042743((4-Chloro-phenyl)-[4-(2-ethyl-5,7-dimethyl-imidazo...)
Affinity DataIC50: 19nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049193(9,28-dipropyl-13-sulfurdioxo-1,14,22,27-tetraazape...)
Affinity DataIC50: 24nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240609(CHEMBL1016 | 2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049192((S)-2-Diphenylacetyl-6-phenyl-1,2,3,4-tetrahydro-i...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Guinea pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003387(2-Ethyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 30nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in guinea pig adrenal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
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