Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50006007
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043717({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.230nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043712({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50009180(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50: 0.280nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50009180(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.670nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.670nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043717({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.870nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043712({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043713(3-{(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 2.24nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043713(3-{(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 2.24nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043713(3-{(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 2.24nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043713(3-{(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 2.24nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043717({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 2.98nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043719(3-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043719(3-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 3.40nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043719(3-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043719(3-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 3.40nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043714({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043716({(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: 4.83nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043716({(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: 4.83nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043716({(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: 4.83nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043716({(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50: 4.83nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043717({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 5.15nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043714({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 6.30nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043715({(4R,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 210nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043715({(4R,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 920nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043712({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043715({(4R,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50009180(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 2.89E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 2.89E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043718((4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 3.30E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043718((4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043718((4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043718((4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 3.30E+3nMAssay Description:In vitro inhibition of electrically induced smooth muscle contractions of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50009180(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043712({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 3.76E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043711(2-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043711(2-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043711(2-(2-{[(4R,10R,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043715({(4R,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 5.50E+3nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043714({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of [3H]CTOP binding to rat brain homogenate mu-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50043714({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 6.80E+4nMAssay Description:In vitro inhibition of electrically evoked contractions in guinea pig ileum longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed