Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50005972
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043244(4'-(1-Methyl-2'-propyl-1H-[2,5']bibenzoimidazolyl-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043260(2-Butyl-6-(1,1-dioxo-1lambda*6*-[1,2]thiazinan-2-y...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043257(6-Imidazo[1,2-a]pyridin-2-yl-4-methyl-2-propyl-1-[...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043246(4'-(6-Imidazo[1,2-a]pyridin-2-yl-4-methyl-2-propyl...)
Affinity DataIC50: 4nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043277(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 4nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043247(4-Methyl-2-propyl-6-pyridin-2-yl-1-[2'-(1H-tetrazo...)
Affinity DataIC50: 5nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043279(1-Methyl-2'-propyl-3'-[2'-(1H-tetrazol-5-yl)-biphe...)
Affinity DataIC50: 5nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043248(3-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 8nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043263(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 10nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043255(2-Propyl-6-pyridin-2-yl-1-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataIC50: 11nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043271(1,7'-Dimethyl-2'-propyl-3'-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043252(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 21nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043269(4'-[2-Butyl-6-(3,3-dimethyl-ureido)-benzoimidazol-...)
Affinity DataIC50: 24nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50035429(4'-[2-Butyl-6-(3-cyclohexyl-ureido)-benzoimidazol-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043268(4'-[2-Butyl-6-(3-cyclohexyl-1-methyl-ureido)-benzo...)
Affinity DataIC50: 26nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043281(4'-{2-Butyl-6-[methyl-(propane-1-sulfonyl)-amino]-...)
Affinity DataIC50: 33nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043249(4'-[2-Butyl-6-(1,1-dioxo-1lambda*6*-[1,2]thiazinan...)
Affinity DataIC50: 34nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50: 35nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043270(4'-[2-Butyl-6-(2-oxo-piperidin-1-yl)-benzoimidazol...)
Affinity DataIC50: 81nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043265(4'-(2-Butyl-6-pentanoylamino-benzoimidazol-1-ylmet...)
Affinity DataIC50: 86nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043275(4'-(6-Dimethylaminomethyl-4-methyl-2-propyl-benzoi...)
Affinity DataIC50: 158nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043256(4'-(2-Butyl-6-piperidin-1-yl-benzoimidazol-1-ylmet...)
Affinity DataIC50: 160nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043276(4'-[2-Butyl-7-(3-cyclohexyl-ureido)-benzoimidazol-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043254(4'-(6-Acetylamino-2-butyl-benzoimidazol-1-ylmethyl...)
Affinity DataIC50: 180nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043245(2-{2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50: 240nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataIC50: 350nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043259(4'-(2-Butyl-6-pentylamino-benzoimidazol-1-ylmethyl...)
Affinity DataIC50: 390nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50005347(CHEMBL7632 | 4'-((2-butyl-1H-benzo[d]imidazol-1-yl...)
Affinity DataIC50: 400nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043273(4'-(5-Acetylamino-2-butyl-benzoimidazol-1-ylmethyl...)
Affinity DataIC50: 460nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043274(4'-(2-Butyl-7-methyl-benzoimidazol-1-ylmethyl)-bip...)
Affinity DataIC50: 480nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043272(4'-(6-Amino-2-butyl-benzoimidazol-1-ylmethyl)-biph...)
Affinity DataIC50: 540nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043266(4'-[2-Butyl-5-(3-cyclohexyl-ureido)-benzoimidazol-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043258(4'-(5-Amino-2-butyl-benzoimidazol-1-ylmethyl)-biph...)
Affinity DataIC50: 820nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043261(4'-(2-Butyl-6-methyl-benzoimidazol-1-ylmethyl)-bip...)
Affinity DataIC50: 850nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043253(4'-(7-Amino-2-butyl-benzoimidazol-1-ylmethyl)-biph...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043267(4'-(2-Butyl-5-methyl-benzoimidazol-1-ylmethyl)-bip...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043278(4'-(2-Butyl-4-methyl-benzoimidazol-1-ylmethyl)-bip...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043262(4'-(4-Amino-2-butyl-benzoimidazol-1-ylmethyl)-biph...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043250(4'-(7-Acetylamino-2-butyl-benzoimidazol-1-ylmethyl...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043264(4'-(4-Acetylamino-2-butyl-benzoimidazol-1-ylmethyl...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor B(Rat)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043251(4'-[2-Butyl-4-(3-cyclohexyl-ureido)-benzoimidazol-...)
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed