Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50005782
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040929(5,6-bis(phenylamino)-1H-isoindole-1,3(2H)-dione | ...)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040930(5,6-Bis-(4-fluoro-phenylamino)-isoindole-1,3-dione...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040917(5-(Methyl-phenyl-amino)-6-phenylamino-isoindole-1,...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040930(5,6-Bis-(4-fluoro-phenylamino)-isoindole-1,3-dione...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040916(5,6-Bis-(4-hydroxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040920(5,6-Bis-p-tolylamino-isoindole-1,3-dione | CHEMBL7...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040920(5,6-Bis-p-tolylamino-isoindole-1,3-dione | CHEMBL7...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040929(5,6-bis(phenylamino)-1H-isoindole-1,3(2H)-dione | ...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040916(5,6-Bis-(4-hydroxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040917(5-(Methyl-phenyl-amino)-6-phenylamino-isoindole-1,...)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM2672(6,7,12,13-Tetrahydro-5,7-dioxo-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50040917(5-(Methyl-phenyl-amino)-6-phenylamino-isoindole-1,...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of PDGF-dependent autophosphorylation of PDGF-R in mouse BALB/c3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040916(5,6-Bis-(4-hydroxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040929(5,6-bis(phenylamino)-1H-isoindole-1,3(2H)-dione | ...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040914(5-(4-Methoxy-phenylamino)-6-phenylamino-isoindole-...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040914(5-(4-Methoxy-phenylamino)-6-phenylamino-isoindole-...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM2583(bis-indolylmaleimide deriv. 8a | 3,4-bis(1H-indol-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040918(5,6-Bis-(methyl-phenyl-amino)-isoindole-1,3-dione ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040923(N-Methyl-4,5-dianilinophthalimide | 2-Methyl-5,6-b...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM2583(bis-indolylmaleimide deriv. 8a | 3,4-bis(1H-indol-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040930(5,6-Bis-(4-fluoro-phenylamino)-isoindole-1,3-dione...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040921(5,6-Bis-(4-diethylamino-phenylamino)-isoindole-1,3...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040912(5,6-Bis-cyclohexylamino-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040921(5,6-Bis-(4-diethylamino-phenylamino)-isoindole-1,3...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040927(N-(1,3-Dioxo-6-phenylamino-2,3-dihydro-1H-isoindol...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040929(5,6-bis(phenylamino)-1H-isoindole-1,3(2H)-dione | ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040930(5,6-Bis-(4-fluoro-phenylamino)-isoindole-1,3-dione...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040912(5,6-Bis-cyclohexylamino-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040925(5,6-Bis-(4-methoxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040923(N-Methyl-4,5-dianilinophthalimide | 2-Methyl-5,6-b...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040918(5,6-Bis-(methyl-phenyl-amino)-isoindole-1,3-dione ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040919(5,6-Bis-(biphenyl-4-ylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040922(2-Phenyl-5,6-bis-phenylamino-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040922(2-Phenyl-5,6-bis-phenylamino-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040925(5,6-Bis-(4-methoxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040927(N-(1,3-Dioxo-6-phenylamino-2,3-dihydro-1H-isoindol...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040913(1,4-Diphenyl-1,2,3,4-tetrahydro-pyrrolo[3,4-g]quin...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040912(5,6-Bis-cyclohexylamino-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040913(1,4-Diphenyl-1,2,3,4-tetrahydro-pyrrolo[3,4-g]quin...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1/ABL2(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040917(5-(Methyl-phenyl-amino)-6-phenylamino-isoindole-1,...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against v-abl tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040915(5,6-Bis-(4-iodo-phenylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040914(5-(4-Methoxy-phenylamino)-6-phenylamino-isoindole-...)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040924(5,6-Bis-phenylsulfanyl-isoindole-1,3-dione | CHEMB...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50040919(5,6-Bis-(biphenyl-4-ylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PDGF-dependent autophosphorylation of PDGF-R in mouse BALB/c3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040931(4,5-Bis-(4-fluoro-phenylamino)-phthalic acid dimet...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040926(4,5-Bis-phenylamino-phthalic acid dimethyl ester |...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040921(5,6-Bis-(4-diethylamino-phenylamino)-isoindole-1,3...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against c-src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50040919(5,6-Bis-(biphenyl-4-ylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EGF-dependent autophosphorylation of EGF-R in human A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50040925(5,6-Bis-(4-methoxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PDGF-dependent autophosphorylation of PDGF-R in mouse BALB/c3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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