Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50036267
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Toledo

Curated by ChEMBL
LigandPNGBDBM50039841(6-Amino-2,3,4,5-tetrahydro-pyridine-4-carboxylic a...)
Affinity DataIC50: 1.20E+5nMAssay Description:Affinity for muscarinic receptor M1 in rat brain was measured by inhibition of [3H](R)-quinuclidinyl benzilate (QNB) bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Toledo

Curated by ChEMBL
LigandPNGBDBM50039836(6-Amino-2,3,4,5-tetrahydro-pyridine-2-carboxylic a...)
Affinity DataIC50: 2.50E+5nMAssay Description:Affinity for muscarinic receptor M1 in rat brain was measured by inhibition of [3H](R)-quinuclidinyl benzilate (QNB) bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
University of Toledo

Curated by ChEMBL
LigandPNGBDBM50039845(2-Amino-3,4,5,6-tetrahydro-pyridine-3-carboxylic a...)
Affinity DataIC50: 3.20E+5nMAssay Description:Affinity for muscarinic receptor M1 in rat brain was measured by inhibition of [3H](R)-quinuclidinyl benzilate (QNB) bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed