Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50005554
Affinity DataEC50: 6.40E+3nMAssay Description:In vitro ability to contract isolated guinea pig ileum was used to estimate M3 agonist effectMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: >5.10E+4nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 83nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]Pirenzepine binding on rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataEC50: >5.10E+4nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: >1.20E+3nMAssay Description:M1 agonist activity estimated by rat superior cervical ganglion depolarizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 680nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 6.50E+3nMAssay Description:In vitro ability to contract isolated guinea pig ileum was used to estimate M2/M3 agonist effectMore data for this Ligand-Target Pair
Affinity DataEC50: 4.40E+3nMAssay Description:In vitro ability to contract isolated guinea pig ileum was used to estimate M2/M3 agonist effectMore data for this Ligand-Target Pair
Affinity DataEC50: 840nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+3nMAssay Description:M1 agonist activity estimated by rat superior cervical ganglion depolarizationMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 640nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair



































