Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 4978
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84628(EC5-21)
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84621(BIM 23042)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82462(D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr-NH2 | BIM 2...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84620(DC23-60)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82462(D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr-NH2 | BIM 2...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-Lys-L-Val-L-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84628(EC5-21)
Affinity DataKi:  0.970nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84621(BIM 23042)
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-Lys-L-Val-L-...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50063819(CHEMBL413535 | BIM 23050 | cyclo[NMeDAla-Tyr-DTrp-...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | NSC_3086456 | MK 678)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  1.54nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  1.55nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | NSC_3086456 | MK 678)
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84623(NC4-28B)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
Affinity DataKi:  2.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84620(DC23-60)
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84623(NC4-28B)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84622(BIM 23057)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
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