Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50005537
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038019(Tyr-Gly-Gly-Phe-D-Leu-Arg-Arg-Ile-Arg-Pro-Lys-NH2 ...)
Affinity DataIC50: 0.530nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataIC50: 0.580nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038020(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-Cys-NH2 ...)
Affinity DataIC50: 0.710nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453445(CHEMBL2112652)
Affinity DataIC50: 1nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038016(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-Pen-NH2 ...)
Affinity DataIC50: 1nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038012(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-Cys-NH2 ...)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038014(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-D-Pen-NH2 ...)
Affinity DataIC50: 2nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038010(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-D-Pen-NH2 ...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038011(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-D-Cys-NH2 ...)
Affinity DataIC50: 3.10nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038014(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-D-Pen-NH2 ...)
Affinity DataIC50: 5nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038020(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-Cys-NH2 ...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038019(Tyr-Gly-Gly-Phe-D-Leu-Arg-Arg-Ile-Arg-Pro-Lys-NH2 ...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038010(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-D-Pen-NH2 ...)
Affinity DataIC50: 7.10nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataIC50: 9.90nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453445(CHEMBL2112652)
Affinity DataIC50: 12nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453445(CHEMBL2112652)
Affinity DataIC50: 14nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038013(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-Cys-NH2 | ...)
Affinity DataIC50: 15nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038007(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-Pen-NH2 | ...)
Affinity DataIC50: 15nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038020(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-Cys-NH2 ...)
Affinity DataIC50: 16nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038016(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-Pen-NH2 ...)
Affinity DataIC50: 17nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038006(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-D-Cys-NH...)
Affinity DataIC50: 18nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038019(Tyr-Gly-Gly-Phe-D-Leu-Arg-Arg-Ile-Arg-Pro-Lys-NH2 ...)
Affinity DataIC50: 19nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038018(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-Cys-NH2 | ...)
Affinity DataIC50: 26nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataIC50: 26nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453446(CHEMBL2369128)
Affinity DataIC50: 27nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038012(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-Cys-NH2 ...)
Affinity DataIC50: 31nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038015(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-Pen-NH2 | ...)
Affinity DataIC50: 43nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038006(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-D-Cys-NH...)
Affinity DataIC50: 51nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038011(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-D-Cys-NH2 ...)
Affinity DataIC50: 68nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038017(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-D-Pen-NH...)
Affinity DataIC50: 71nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038009(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-Pen-NH2 ...)
Affinity DataIC50: 87nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038009(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-Pen-NH2 ...)
Affinity DataIC50: 87nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453446(CHEMBL2369128)
Affinity DataIC50: 96nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038015(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-Pen-NH2 | ...)
Affinity DataIC50: 99nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038021(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-D-Pen-NH...)
Affinity DataIC50: 100nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038008(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-D-Cys-NH...)
Affinity DataIC50: 104nMAssay Description:Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038021(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-D-Pen-NH...)
Affinity DataIC50: 108nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038013(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-Cys-NH2 | ...)
Affinity DataIC50: 116nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038008(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-D-Cys-NH...)
Affinity DataIC50: 128nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038018(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-Cys-NH2 | ...)
Affinity DataIC50: 224nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038010(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-D-Pen-NH2 ...)
Affinity DataIC50: 232nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038012(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-Cys-NH2 ...)
Affinity DataIC50: 242nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038014(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-D-Pen-NH2 ...)
Affinity DataIC50: 245nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038016(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-Pen-NH2 ...)
Affinity DataIC50: 319nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038006(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-D-Cys-NH...)
Affinity DataIC50: 390nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038007(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-Pen-NH2 | ...)
Affinity DataIC50: 473nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038017(Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-Arg-Pro-D-Pen-NH...)
Affinity DataIC50: 563nMAssay Description:Binding affinity at mu opioid receptor in guinea pig brain by [3H]DAMGO displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038011(Tyr-Gly-Gly-Phe-Pen-Arg-Arg-Ile-Arg-Pro-D-Cys-NH2 ...)
Affinity DataIC50: 717nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038007(Tyr-Gly-Gly-Phe-Cys-Arg-Arg-Ile-Arg-Pro-Pen-NH2 | ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50038008(Tyr-Gly-Gly-Phe-D-Cys-Arg-Arg-Ile-Arg-Pro-D-Cys-NH...)
Affinity DataIC50: 1.03E+3nMAssay Description:Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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