Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50005343
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035820(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37830)
Affinity DataIC50: 0.450nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035832(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL35471)
Affinity DataIC50: 1.80nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035825(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL34554)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035829(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34853)
Affinity DataIC50: 30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035834(Ac-Trp-L-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL287753)
Affinity DataIC50: 50nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035833(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37984)
Affinity DataIC50: 70nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035822(Ac-Trp-L-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL37983)
Affinity DataIC50: 300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035823(Ac-Trp-Pro-Asp-Phe-NH2 | Ac-Trp-D-Pro-Asp-Phe-NH2 ...)
Affinity DataIC50: 600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035828(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37900)
Affinity DataIC50: 600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035821(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34916)
Affinity DataIC50: 800nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035828(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37900)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested for binding affinity towards Cholecystokinin type A receptor by measuring its ability to displace [125I]BH-CCK-8 from rat pancrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035823(Ac-Trp-Pro-Asp-Phe-NH2 | Ac-Trp-D-Pro-Asp-Phe-NH2 ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035825(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL34554)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035820(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37830)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035833(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37984)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035831(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL290444)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035836((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035826((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035829(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34853)
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035822(Ac-Trp-L-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL37983)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035835(Trp-D-4-MPt(Me)-Asp-Phe-NH2 | CHEMBL285756)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035836((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035831(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL290444)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPt(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPc(Me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPt(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPc(Me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035834(Ac-Trp-L-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL287753)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50453646(CHEMBL2114402)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035835(Trp-D-4-MPt(Me)-Asp-Phe-NH2 | CHEMBL285756)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035819(Ac-Trp-D-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL37786)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035830(Ac-Trp-D-Nle(Me)-Asp-Phe-NH2 | CHEMBL35394)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035824(Ac-Trp-D-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL285051)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035830(Ac-Trp-D-Nle(Me)-Asp-Phe-NH2 | CHEMBL35394)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035832(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL35471)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035826((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035824(Ac-Trp-D-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL285051)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035821(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34916)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035819(Ac-Trp-D-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL37786)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPt(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPc(Me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPt(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPc(Me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50453646(CHEMBL2114402)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed