Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50005322
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035540(5-(4-tert-Butyl-phenyl)-2,3-dihydro-imidazo[2,1-a]...)
Affinity DataIC50: 900nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035570(5-(4-Thiomorpholin-4-ylmethyl-phenyl)-2,3-dihydro-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035557(5-[4-(2-Methyl-piperidin-1-ylmethyl)-phenyl]-2,3-d...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035548(5-(4-tert-Butyl-phenyl)-8-chloro-2,3-dihydro-imida...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035556(5-(4-Morpholin-4-ylmethyl-phenyl)-2,3-dihydro-imid...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035560(5-Biphenyl-4-yl-2,3-dihydro-imidazo[2,1-a]isoquino...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035539(5-(3-tert-Butyl-phenyl)-2,3-dihydro-imidazo[2,1-a]...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035555(5-p-Tolyl-2,3-dihydro-imidazo[2,1-a]isoquinoline |...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035547(5-(3-Chloro-phenyl)-2,3-dihydro-imidazo[2,1-a]isoq...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035558(5-(2-Fluoro-phenyl)-2,3-dihydro-imidazo[2,1-a]isoq...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035550(5-(4-Ethyl-phenyl)-2,3-dihydro-imidazo[2,1-a]isoqu...)
Affinity DataIC50: 6.30E+3nMAssay Description:Compound were tested for the inhibition of [3H]PAF binding to human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035569(5-(4-Trimethylsilanyl-phenyl)-2,3-dihydro-imidazo[...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035568(4-(2,3-Dihydro-imidazo[2,1-a]isoquinolin-5-yl)-phe...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035554(5-(4-Piperidin-1-ylmethyl-phenyl)-2,3-dihydro-imid...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035553(5-(2-Chloro-phenyl)-2,3-dihydro-imidazo[2,1-a]isoq...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035542(Diallyl-[4-(2,3-dihydro-imidazo[2,1-a]isoquinolin-...)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035544(5-Phenyl-2,3-dihydro-imidazo[2,1-a]isoquinoline | ...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035559(Dicyclohexyl-[4-(2,3-dihydro-imidazo[2,1-a]isoquin...)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035564(5-(4-Fluoro-phenyl)-2,3-dihydro-imidazo[2,1-a]isoq...)
Affinity DataIC50: 1.42E+4nMAssay Description:Compound were tested for the inhibition of [3H]PAF binding to human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035566(5-Thiophen-2-yl-2,3-dihydro-imidazo[2,1-a]isoquino...)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035565(5-(3,4-Dichloro-phenyl)-2,3-dihydro-imidazo[2,1-a]...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035543(5-Benzo[1,3]dioxol-5-yl-2,3-dihydro-imidazo[2,1-a]...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035552(5-(3-Trifluoromethyl-phenyl)-2,3-dihydro-imidazo[2...)
Affinity DataIC50: 1.92E+4nMAssay Description:Compound were tested for the inhibition of [3H]PAF binding to human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035562(5-(3,4-Dimethoxy-phenyl)-2,3-dihydro-imidazo[2,1-a...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035549(5-(4-tert-Butyl-phenyl)-9-methyl-2,3-dihydro-imida...)
Affinity DataIC50: 3.18E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035563(5-(4-Chloro-phenyl)-2,3-dihydro-imidazo[2,1-a]isoq...)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035546(5-(4-tert-Butyl-phenyl)-9-chloro-2,3-dihydro-imida...)
Affinity DataIC50: 4.04E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035537(5-Pyridin-4-yl-2,3-dihydro-imidazo[2,1-a]isoquinol...)
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035541(5-(4-Methoxy-phenyl)-2,3-dihydro-imidazo[2,1-a]iso...)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035545(5-(4-Pyrrolidin-1-ylmethyl-phenyl)-2,3-dihydro-imi...)
Affinity DataIC50: 5.94E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035551(5-(2,4-Dichloro-phenyl)-2,3-dihydro-imidazo[2,1-a]...)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035561(5-(3,4,5-Trimethoxy-phenyl)-2,3-dihydro-imidazo[2,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035567(5-Pyridin-3-yl-2,3-dihydro-imidazo[2,1-a]isoquinol...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50035538(5-Furan-2-yl-2,3-dihydro-imidazo[2,1-a]isoquinolin...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]PAF binding to human platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed