Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 4879
TargetMuscarinic acetylcholine receptor M2(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  1.58nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  6.41nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  33.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  38.0nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM82423(NSC_132947 | CAS_132947 | TRIPITRAMINE)
Affinity DataKi:  38.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  277nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Pisa

Curated by PDSP Ki Database
LigandPNGBDBM50064176(METHOCTRAMINE | N,N''-Bis-[6-(2-methoxy-benzylamin...)
Affinity DataKi:  313nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed