Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50005308
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50035468(NSC-115290 | 4-(4-Hydroxy-9,10-dioxo-9,10-dihydro-...)
Affinity DataKi:  7.80E+3nMAssay Description:Binding affinity with protein kinase C (PK-C) alpha bound to labeled [20-3H]-PDBU at a conc of 30 ug/mLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50035469(2-hydroxy-1-(2-hydroxy-1-phenylcarbonyloxyethyl)-3...)
Affinity DataKi:  1.29E+4nMAssay Description:Binding affinity with protein kinase C (PK-C) alpha bound to labeled [20-3H]-PDBU at a conc of 30 ug/mLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50035466(2-[1-[Bis-(2-hydroxy-ethyl)-amino]-meth-(Z)-yliden...)
Affinity DataKi:  1.61E+4nMAssay Description:Binding affinity with protein kinase C (PK-C) alpha bound to labeled [20-3H]-PDBU at a conc of 30 ug/mLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50035467(3-(4-Hydroxy-9,10-dioxo-9,10-dihydro-anthracen-1-y...)
Affinity DataKi:  2.66E+4nMAssay Description:Binding affinity with protein kinase C (PK-C) alpha bound to labeled [20-3H]-PDBU at a conc of 30 ug/mLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50035470(Acetic acid 2-((1S,2R,4aR,5S,8aR)-6-acetoxy-5-acet...)
Affinity DataKi:  3.77E+4nMAssay Description:Binding affinity with protein kinase C (PK-C) alpha bound to labeled [20-3H]-PDBU at a conc of 30 ug/mLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed