Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50005239
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034722((Z)-Octadec-9-enoic acid (1,2-diphenyl-ethyl)-amid...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034738(3-(Decyl-dimethyl-silanyl)-N-(1-phenyl-2-p-tolyl-e...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034719(N-[2-(4-Acetylamino-phenyl)-1-phenyl-ethyl]-2,2-di...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034739((Z)-Octadec-9-enoic acid [2-(4-amino-phenyl)-1-phe...)
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034741(N-[2-(4-Methanesulfonylamino-phenyl)-1-phenyl-ethy...)
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034737(N-(1,2-Diphenyl-ethyl)-2,2-diphenyl-acetamide | CH...)
Affinity DataIC50: 460nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034720(N-[2-(3,4-Dimethoxy-phenyl)-1-phenyl-ethyl]-2,2-di...)
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034725(N-[2-(4-Hydroxy-phenyl)-1-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50028868(N-[2-(4-Amino-phenyl)-1-phenyl-ethyl]-2,2-diphenyl...)
Affinity DataIC50: 900nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034732(N-[1-(4-Hydroxy-phenyl)-2-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034716(N-[1-(4-Methoxy-phenyl)-2-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034723(N-[1-(3-Methoxy-phenyl)-2-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034740(N-[2-(4-Methoxy-phenyl)-1-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50028868(N-[2-(4-Amino-phenyl)-1-phenyl-ethyl]-2,2-diphenyl...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034721(N-[1-(2-Methoxy-phenyl)-2-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034731(2,2-Diphenyl-N-(1-phenyl-2-pyridin-4-yl-ethyl)-ace...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034734(2,2-Diphenyl-N-(2-phenyl-1-pyridin-4-yl-ethyl)-ace...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034742(N-[2-(4-Methoxy-phenyl)-1-(3-methoxy-phenyl)-ethyl...)
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034726(N-[1-(4-Amino-phenyl)-2-phenyl-ethyl]-2,2-diphenyl...)
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50022279(CL-277082 | 3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dime...)
Affinity DataIC50: 3.20E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034730(N-(2-Imidazol-1-yl-1-phenyl-ethyl)-2,2-diphenyl-ac...)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034733(2,2-Diphenyl-N-(2-phenyl-1-pyridin-3-yl-ethyl)-ace...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034727(N-[2-(3-Amino-phenyl)-1-phenyl-ethyl]-2,2-diphenyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034729(N-[2-(1-Heptyl-1H-imidazol-2-yl)-1-phenyl-ethyl]-2...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034714(2,2-Diphenyl-N-{1-phenyl-2-[1-(2-trimethylsilanyl-...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50005944(2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034736(2,2-Diphenyl-N-{2-phenyl-1-[1-(2-trimethylsilanyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034735(N-[1-(1-Oxy-pyridin-4-yl)-2-phenyl-ethyl]-2,2-diph...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034728(4-(1-Diphenylacetylamino-2-phenyl-ethyl)-benzoic a...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034724(4-(2-Diphenylacetylamino-2-phenyl-ethyl)-benzoic a...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034718(N-[1-(1H-Imidazol-2-yl)-2-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034717(N-[2-(1H-Imidazol-2-yl)-1-phenyl-ethyl]-2,2-diphen...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034715(4-(2-Diphenylacetylamino-2-phenyl-ethyl)-benzoic a...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50034743(N-[1,2-Bis-(4-methoxy-phenyl)-ethyl]-2,2-diphenyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed