Compile Data Set for Download or QSAR
Report error Found 118 Enz. Inhib. hit(s) with all data for entry = 50005229
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.00150nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034581(Peptide boronate | CHEMBL36744)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034581(Peptide boronate | CHEMBL36744)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.00490nMAssay Description:Binding affinity against kallikreinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034574(Peptide boronate | CHEMBL288150)
Affinity DataKi:  0.00700nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(Peptide boronate | CHEMBL290577)
Affinity DataKi:  0.00700nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(Peptide boronate | CHEMBL285285)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(Peptide boronate | CHEMBL285285)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(Peptide boronate | CHEMBL285285)
Affinity DataKi:  0.0180nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(Peptide boronate | CHEMBL291026)
Affinity DataKi:  0.0190nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(Peptide boronate | CHEMBL291026)
Affinity DataKi:  0.0190nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(Peptide boronate | CHEMBL418050)
Affinity DataKi:  0.0210nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(Peptide boronate | CHEMBL290577)
Affinity DataKi:  0.0240nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034583(Peptide boronate | CHEMBL287918)
Affinity DataKi:  0.0270nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034574(Peptide boronate | CHEMBL288150)
Affinity DataKi:  0.0280nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034573(Peptide boronate | CHEMBL291261)
Affinity DataKi:  0.0280nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034573(Peptide boronate | CHEMBL291261)
Affinity DataKi:  0.0340nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034583(Peptide boronate | CHEMBL287918)
Affinity DataKi:  0.0420nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034581(Peptide boronate | CHEMBL36744)
Affinity DataKi:  0.0540nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(Peptide boronate | CHEMBL418050)
Affinity DataKi:  0.0590nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034576(Peptide boronate | CHEMBL288176)
Affinity DataKi:  0.0820nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(Peptide boronate | CHEMBL291026)
Affinity DataKi:  0.115nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(Peptide boronate | CHEMBL418050)
Affinity DataKi:  0.130nMAssay Description:Binding affinity against alpha thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034576(Peptide boronate | CHEMBL288176)
Affinity DataKi:  0.140nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(Peptide boronate | CHEMBL285285)
Affinity DataKi:  0.150nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(Peptide boronate | CHEMBL290577)
Affinity DataKi:  0.152nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin G(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(Peptide boronate | CHEMBL418050)
Affinity DataKi:  0.174nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin G(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(Peptide boronate | CHEMBL285285)
Affinity DataKi:  0.187nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(Peptide boronate | CHEMBL290577)
Affinity DataKi:  0.270nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(Peptide boronate | CHEMBL291026)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(Peptide boronate | CHEMBL290577)
Affinity DataKi:  0.365nMAssay Description:Binding affinity towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034580(Peptide boronate | CHEMBL418050)
Affinity DataKi:  0.440nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034583(Peptide boronate | CHEMBL287918)
Affinity DataKi:  0.450nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034573(Peptide boronate | CHEMBL291261)
Affinity DataKi:  0.560nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034577(Peptide boronate | CHEMBL291026)
Affinity DataKi:  0.580nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034574(Peptide boronate | CHEMBL288150)
Affinity DataKi:  0.670nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against Urokinase plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity towards porcine pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against gamma thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin G(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  0.848nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin G(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034579(Peptide boronate | CHEMBL290577)
Affinity DataKi:  0.916nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034582(Peptide boronate | CHEMBL2448441)
Affinity DataKi:  1nMAssay Description:Binding affinity against thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034585(Peptide boronate | CHEMBL285285)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034583(Peptide boronate | CHEMBL287918)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034574(Peptide boronate | CHEMBL288150)
Affinity DataKi:  1.21nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50034576(Peptide boronate | CHEMBL288176)
Affinity DataKi:  1.46nMAssay Description:Binding affinity against ChymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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