Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50005053
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031962(3-(5,7-Dimethyl-2-propyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataKi:  0.290nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031954(3-(2-Cyclopropyl-5,7-dimethyl-imidazo[4,5-b]pyridi...)
Affinity DataKi:  0.450nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031953(3-(2-Ethyl-6-methoxy-[1,5]naphthyridin-4-yloxymeth...)
Affinity DataKi:  0.480nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031957(5,7-Dimethyl-2-propyl-3-[11-(1H-tetrazol-5-yl)-5H-...)
Affinity DataKi:  0.490nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031960(3-(2-Ethyl-quinolin-4-yloxymethyl)-11-(1H-tetrazol...)
Affinity DataKi:  0.650nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031961(3-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-yl...)
Affinity DataKi:  0.660nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031955(5,7-Dimethyl-2-propyl-3-[11-(1H-tetrazol-5-yl)-dib...)
Affinity DataKi:  0.700nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031964(3-[(5-Ethyl-pyrazolo[1,5-a]pyrimidin-7-ylamino)-me...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031956(3-(2-Ethyl-5,6,7,8-tetrahydro-quinolin-4-yloxymeth...)
Affinity DataKi:  1.30nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031959(2-Butyl-5-chloro-3-[5-oxo-11-(1H-tetrazol-5-yl)-5H...)
Affinity DataKi:  2.10nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031965(2-Ethyl-4-[5-oxo-11-(1H-tetrazol-5-yl)-5H-dibenzo[...)
Affinity DataKi:  2.70nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031966(2-Ethoxy-3-[5-oxo-11-(1H-tetrazol-5-yl)-5H-dibenzo...)
Affinity DataKi:  2.70nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031950(2,6-Dimethyl-4-{[5-oxo-11-(1H-tetrazol-5-yl)-5H-di...)
Affinity DataKi:  2.90nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031951(2-Ethoxy-3-[11-(1H-tetrazol-5-yl)-dibenzo[b,f]oxep...)
Affinity DataKi:  3.90nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031963(2,6-Dimethyl-4-[5-oxo-11-(1H-tetrazol-5-yl)-5H-dib...)
Affinity DataKi:  4.30nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031949(3-(2-Methyl-5,6,7,8-tetrahydro-quinolin-4-yloxymet...)
Affinity DataKi:  4.30nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031952((S)-3-Methyl-2-{[5-oxo-11-(1H-tetrazol-5-yl)-5H-di...)
Affinity DataKi:  8.70nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031958((S)-3-Methyl-2-{pentanoyl-[11-(1H-tetrazol-5-yl)-d...)
Affinity DataKi:  9.60nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50031948(2-Butyl-5-chloro-3-[5-oxo-11-(1H-tetrazol-5-yl)-5H...)
Affinity DataKi:  12nMAssay Description:Ability to displace [125I]AII binding to COS cells transfected with a cDNA encoding human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed