Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50036373
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031297(7-(3-{4-[Bis-(4-fluoro-phenyl)-methyl]-piperazin-1...)
Affinity DataIC50: 38nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031296(7-[3-(4-Benzhydryl-piperidin-1-yl)-propyl]-1,3-dim...)
Affinity DataIC50: 40nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031296(7-[3-(4-Benzhydryl-piperidin-1-yl)-propyl]-1,3-dim...)
Affinity DataIC50: 41nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031297(7-(3-{4-[Bis-(4-fluoro-phenyl)-methyl]-piperazin-1...)
Affinity DataIC50: 43nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031296(7-[3-(4-Benzhydryl-piperidin-1-yl)-propyl]-1,3-dim...)
Affinity DataIC50: 44nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM22873(Bactil | CHEMBL305660 | 1-(4-tert-butylphenyl)-4-[...)
Affinity DataIC50: 45nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031296(7-[3-(4-Benzhydryl-piperidin-1-yl)-propyl]-1,3-dim...)
Affinity DataIC50: 46nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM22873(Bactil | CHEMBL305660 | 1-(4-tert-butylphenyl)-4-[...)
Affinity DataIC50: 47nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM22873(Bactil | CHEMBL305660 | 1-(4-tert-butylphenyl)-4-[...)
Affinity DataIC50: 61nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50017376(1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylmethyl...)
Affinity DataIC50: 94nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031297(7-(3-{4-[Bis-(4-fluoro-phenyl)-methyl]-piperazin-1...)
Affinity DataIC50: 220nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031297(7-(3-{4-[Bis-(4-fluoro-phenyl)-methyl]-piperazin-1...)
Affinity DataIC50: 670nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM22873(Bactil | CHEMBL305660 | 1-(4-tert-butylphenyl)-4-[...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031297(7-(3-{4-[Bis-(4-fluoro-phenyl)-methyl]-piperazin-1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM22873(Bactil | CHEMBL305660 | 1-(4-tert-butylphenyl)-4-[...)
Affinity DataIC50: 1.10E+3nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50017376(1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylmethyl...)
Affinity DataIC50: 2.90E+3nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50031296(7-[3-(4-Benzhydryl-piperidin-1-yl)-propyl]-1,3-dim...)
Affinity DataIC50: 7.30E+3nMAssay Description:Compound is evaluated for in vitro receptor binding affinity against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed