Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50036234
TargetMu-type opioid receptor(Bovine)
Institute

Curated by ChEMBL
LigandPNGBDBM50030143(bis-(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azape...)
Affinity DataIC50: 0.400nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGO radiolabeled opioidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
Institute

Curated by ChEMBL
LigandPNGBDBM50030144(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacy...)
Affinity DataIC50: 0.630nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
Institute

Curated by ChEMBL
LigandPNGBDBM50030145(bis-(1N-[4-cyclopropylmethyl-10-hydroxy-14-oxo-12-...)
Affinity DataIC50: 3.30nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGO radiolabeled opioidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50030145(bis-(1N-[4-cyclopropylmethyl-10-hydroxy-14-oxo-12-...)
Affinity DataIC50: 10nMAssay Description:Evaluation for the inhibition of kappa opioid binding to bovine striatal membranes by the affinity ligand 1 nM [3H]U-69593 radiolabeled opioidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50030143(bis-(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azape...)
Affinity DataIC50: 11nMAssay Description:Evaluation for the inhibition of delta opioid binding to bovine striatal membranes by the affinity ligand 0.2 nM [3H]-p-Cl-DPDPE radiolabeled opioidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50030144(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacy...)
Affinity DataIC50: 12nMAssay Description:Evaluation for the inhibition of delta opioid binding to bovine striatal membranes by the affinity ligand 0.2 nM [3H]p-Cl-DPDPEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50030145(bis-(1N-[4-cyclopropylmethyl-10-hydroxy-14-oxo-12-...)
Affinity DataIC50: 24nMAssay Description:Evaluation for the inhibition of delta opioid binding to bovine striatal membranes by the affinity ligand 0.2 nM [3H]-p-Cl-DPDPE radiolabeled opioidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50030144(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacy...)
Affinity DataIC50: 41nMAssay Description:Evaluation for the inhibition of kappa opioid binding to bovine striatal membranes by the affinity ligand 1 nM [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Institute

Curated by ChEMBL
LigandPNGBDBM50030143(bis-(1N-[10-hydroxy-4-methyl-14-oxo-12-oxa-4-azape...)
Affinity DataIC50: 41nMAssay Description:Evaluation for the inhibition of kappa opioid binding to bovine striatal membranes by the affinity ligand 1 nM [3H]-U-69,593 radiolabeled opioidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed