Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50048617
LigandChemical structure of BindingDB Monomer ID 50029050BDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataKi:  200nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50029051BDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataKi:  500nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223426BDBM50223426(CHEBI:10304 | Corbadrine | Levonordefrin | Neo-Cob...)
Affinity DataKi:  3.60E+3nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223426BDBM50223426(CHEBI:10304 | Corbadrine | Levonordefrin | Neo-Cob...)
Affinity DataKi:  7.30E+3nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223492BDBM50223492(CHEMBL2114304)
Affinity DataKi:  1.10E+4nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223427BDBM50223427(Dioxifedrine)
Affinity DataKi:  2.80E+4nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223425BDBM50223425(CHEMBL23040)
Affinity DataKi:  1.46E+5nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223426BDBM50223426(CHEBI:10304 | Corbadrine | Levonordefrin | Neo-Cob...)
Affinity DataKi:  2.32E+6nMAssay Description:Compound was evaluated for inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat forebrain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2018
Entry Details Article
PubMed