Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50035500
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 3nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-2 adrenergic receptor in calf lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 4.90nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026852(1-Isopropylamino-3-(7-methyl-indan-4-yloxy)-propan...)
Affinity DataIC50: 18nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-2 adrenergic receptor in calf lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50367112(CHEMBL1788270)
Affinity DataIC50: 20nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-2 adrenergic receptor in calf lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026853(Fluoren-9-one O-(3-tert-butylamino-2-hydroxy-propy...)
Affinity DataIC50: 25nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-2 adrenergic receptor in calf lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50367111(CHEMBL305153)
Affinity DataIC50: 29nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50367111(CHEMBL305153)
Affinity DataIC50: 31nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-2 adrenergic receptor in calf lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50405521(ALO 1401-02 | ALO-1401-02 | Betaxolol | BETAXOLOL ...)
Affinity DataIC50: 37nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50026853(Fluoren-9-one O-(3-tert-butylamino-2-hydroxy-propy...)
Affinity DataIC50: 38nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50367112(CHEMBL1788270)
Affinity DataIC50: 43nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50026852(1-Isopropylamino-3-(7-methyl-indan-4-yloxy)-propan...)
Affinity DataIC50: 186nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-1 adrenergic receptor in dog heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50405521(ALO 1401-02 | ALO-1401-02 | Betaxolol | BETAXOLOL ...)
Affinity DataIC50: 657nMAssay Description:Compound was tested for inhibition of [3H]dihydroalprenolol radioligand binding to Beta-2 adrenergic receptor in calf lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed