Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 4799
TargetNorepinephrine transporter(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50022784(Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxe...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetNorepinephrine transporter(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  16.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetHistamine H1 receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  360nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM50022784(Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxe...)
Affinity DataKi:  750nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetHistamine H1 receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  880nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM50022784(Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxe...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  1.75E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetHistamine H1 receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM82084(CAS_62373-97-1 | LR 5182 | EW5182)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  2.45E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  4.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+/-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquin...)
Affinity DataKi:  6.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetHistamine H1 receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50022784(Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxe...)
Affinity DataKi:  6.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  9.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
LigandPNGBDBM50022784(Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxe...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50022784(Methyl-(3-phenyl-3-o-tolyloxy-propyl)-amine(tomoxe...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetHistamine H1 receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+/-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquin...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM82084(CAS_62373-97-1 | LR 5182 | EW5182)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2011
Entry Details
PubMed