Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50034922
TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 1.10nMAssay Description:Tested for the inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane(CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 6nMAssay Description:Tested for the inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane(CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50450461(CHEMBL2367718)
Affinity DataIC50: 13nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291421((S)-3-{(S)-2-[(1S,2S)-2-Benzyloxycarbonylamino-1-c...)
Affinity DataIC50: 15nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 25nMAssay Description:Tested for the inhibition of specific [3H]propionyl-CCK-8 binding to guinea pig pancreatic Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291428(2-{2-[(S)-2-((S)-Benzyloxycarbonylamino)-1-cyano-3...)
Affinity DataIC50: 45nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50011197(CHEMBL169054 | 3-{2-[2-tert-Butoxycarbonylamino-3-...)
Affinity DataIC50: 65nMAssay Description:Tested for the inhibition of specific [3H]propionyl-CCK-8 binding to guinea pig pancreatic Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291423((S)-3-{(1R,2S)-2-[(S)-2-tert-Butoxycarbonylamino-3...)
Affinity DataIC50: 180nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291425(2-{2-[(S)-2-((S)-Benzyloxycarbonylamino)-1-cyano-3...)
Affinity DataIC50: 189nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291426((R)-2-((R)-2-Benzyloxycarbonylamino-1-cyano-3-(S)-...)
Affinity DataIC50: 272nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291429((S)-3-[(1S,2S)-2-Benzyloxycarbonylamino-1-cyano-3-...)
Affinity DataIC50: 344nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291428(2-{2-[(S)-2-((S)-Benzyloxycarbonylamino)-1-cyano-3...)
Affinity DataIC50: 483nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291427((S)-3-[(1R,2S)-2-Benzyloxycarbonylamino-1-cyano-3-...)
Affinity DataIC50: 719nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291431((S)-3-{(1S,2S)-2-[(S)-2-tert-Butoxycarbonylamino-3...)
Affinity DataIC50: 920nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291425(2-{2-[(S)-2-((S)-Benzyloxycarbonylamino)-1-cyano-3...)
Affinity DataIC50: 938nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291424((S)-3-{(S)-2-[(1R,2S)-2-Benzyloxycarbonylamino-1-c...)
Affinity DataIC50: 953nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50450461(CHEMBL2367718)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291421((S)-3-{(S)-2-[(1S,2S)-2-Benzyloxycarbonylamino-1-c...)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 1.80E+3nMAssay Description:Tested for the inhibition of specific [3H]propionyl-CCK-8 binding to guinea pig cortical Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291424((S)-3-{(S)-2-[(1R,2S)-2-Benzyloxycarbonylamino-1-c...)
Affinity DataIC50: 3.85E+3nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50011197(CHEMBL169054 | 3-{2-[2-tert-Butoxycarbonylamino-3-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Tested for the inhibition of specific [3H]propionyl-CCK-8 binding to guinea pig cortical Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291430([(1S,2R)-2-((S)-1-Carbamoyl-2-phenyl-ethylamino)-2...)
Affinity DataIC50: 5.22E+3nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291430([(1S,2R)-2-((S)-1-Carbamoyl-2-phenyl-ethylamino)-2...)
Affinity DataIC50: 5.22E+3nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291426((R)-2-((R)-2-Benzyloxycarbonylamino-1-cyano-3-(S)-...)
Affinity DataIC50: 8.63E+3nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291431((S)-3-{(1S,2S)-2-[(S)-2-tert-Butoxycarbonylamino-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291422([(1S,2S)-2-((S)-1-Carbamoyl-2-phenyl-ethylamino)-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291429((S)-3-[(1S,2S)-2-Benzyloxycarbonylamino-1-cyano-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291427((S)-3-[(1R,2S)-2-Benzyloxycarbonylamino-1-cyano-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291423((S)-3-{(1R,2S)-2-[(S)-2-tert-Butoxycarbonylamino-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291422([(1S,2S)-2-((S)-1-Carbamoyl-2-phenyl-ethylamino)-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat pancreas membrane Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291430([(1S,2R)-2-((S)-1-Carbamoyl-2-phenyl-ethylamino)-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50291430([(1S,2R)-2-((S)-1-Carbamoyl-2-phenyl-ethylamino)-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific [3H]propionyl-CCK-8 binding to rat cerebral cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article