Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50034865
TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKon:  0.000333M-1s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50093799((R)-1-Amino-13-ethylidene-8,8,11-trimethyl-6-aza-t...)
Affinity DataKoff:  0.0130s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKon:  0.000367M-1s-1 Koff:  0.0155s-1Assay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKoff:  0.0570s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKoff:  0.0567s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50093799((R)-1-Amino-13-ethylidene-8,8,11-trimethyl-6-aza-t...)
Affinity DataKon:  0.000217M-1s-1Assay Description:Kinetic constant for inhibition of fetal bovine serum acetylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKi:  5.90nMAssay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50342601(Huperzine A | CHEMBL1255901)
Affinity DataKi:  5.90nMAssay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetAcetylcholinesterase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50093799((R)-1-Amino-13-ethylidene-8,8,11-trimethyl-6-aza-t...)
Affinity DataKi:  17nMAssay Description:Dissociation constant for the inhibition of fetal bovine serum acetylcholinesterase was determined..More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article