Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50034825
TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286606((4aS,12bR)-11-Chloro-10-hydroxy-4,4,4a,12b-tetrame...)
Affinity DataIC50: 300nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50276581((+/-)-wiedendiol B | CHEMBL456619)
Affinity DataIC50: 600nMAssay Description:Compound was tested for CETP inhibition by a precipitation method to separate lipoproteins after incubation of radiolabeled HDL with LDL and CETP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285079(4-Methoxy-3-((S)-2,5,5,8a-tetramethyl-3,4,4a,5,6,7...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested for CETP inhibition by a precipitation method to separate lipoproteins after incubation of radiolabeled HDL with LDL and CETP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50276581((+/-)-wiedendiol B | CHEMBL456619)
Affinity DataIC50: 5.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285079(4-Methoxy-3-((S)-2,5,5,8a-tetramethyl-3,4,4a,5,6,7...)
Affinity DataIC50: 5.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50240865(CHEMBL157844 | (4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,...)
Affinity DataIC50: 6.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286611(5,5,9,10-tetramethyl-18-oxatetracyclo[8.8.0.01,6.0...)
Affinity DataIC50: 2.20E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286609(1-((4aS,12bR)-9,10-Diacetyl-4,4,4a,12b-tetramethyl...)
Affinity DataIC50: 2.30E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50242257(2-(1,2,4a,5-Tetramethyl-1,2,3,4,4a,7,8,8a-octahydr...)
Affinity DataIC50: 2.50E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286610(13-methoxy-5,5,9,10-tetramethyl-18-oxatetracyclo[8...)
Affinity DataIC50: 4.60E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50240866((-)-ilimaquinone | Ilimaquinone | 2-Hydroxy-5-meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286608(Sulfircin analogue | Sulfuric acid mono-[(1S,2R)-5...)
Affinity DataIC50: 1.90E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholesteryl ester transfer protein(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286607(CHEMBL156156 | (3bR,5aR,6S,7S,9aR,9bR)-7-Hydroxy-6...)
Affinity DataIC50: 1.96E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article