Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50034729
TargetAngiotensin-converting enzyme(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataIC50: 30nMAssay Description:Compound was tested for inhibitory activity against Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetThermolysin(Bacillus thermoproteolyticus)
TBA

Curated by ChEMBL
LigandPNGBDBM50035235(N-[1-(Carbamoylmethyl-carbamoyl)-ethyl]-N''-hydrox...)
Affinity DataIC50: 64nMAssay Description:Compound was tested in vitro for inhibitory activity against thermolysinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50251742((S)-2-{(R)-2-[Hydroxy-((2R,3R,4R,5R,6S)-3,4,5-trih...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280860((S)-2-((S)-2-Benzyloxycarbonylamino-3-mercapto-pro...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280859((S)-3-(1H-Indol-3-yl)-2-(2-mercaptomethyl-4-methyl...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280866((S)-2-(2-Hydroxycarbamoyl-4-methyl-pentanoylamino)...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280861((S)-2-((R)-2-Benzyloxycarbonylamino-3-mercapto-pro...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280862(2-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-mercapto-...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280864((S)-2-[2-((R)-Benzyloxycarbonylamino)-3-mercapto-p...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280858((S)-3-(1H-Indol-3-yl)-2-((R)-2-mercapto-4-methyl-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280863((S)-3-(1H-Indol-3-yl)-2-((S)-2-mercapto-4-methyl-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of putative Endothelin-converting enzyme partially purified from rabbit lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article