Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50030210
TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292475(hypophyllanthin | CHEMBL510130)
Affinity DataIC50: 4.00E+4nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292476(nirtetralin | CHEMBL453822)
Affinity DataIC50: 7.50E+4nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292478((2S,4S)-5,8-dimethoxy-6-methyl-4-phenyl-1,2,3,4-te...)
Affinity DataIC50: 1.60E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50292476(nirtetralin | CHEMBL453822)
Affinity DataIC50: 4.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from ETA receptor in rat A10 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292477(phyllanthin | CHEMBL453568)
Affinity DataIC50: 5.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292476(nirtetralin | CHEMBL453822)
Affinity DataIC50: 5.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292475(hypophyllanthin | CHEMBL510130)
Affinity DataIC50: 5.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50292475(hypophyllanthin | CHEMBL510130)
Affinity DataIC50: 5.80E+5nMAssay Description:Displacement of [125I]endothelin-1 from ETA receptor in rat A10 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50292477(phyllanthin | CHEMBL453568)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [125I]endothelin-1 from ETA receptor in rat A10 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50292477(phyllanthin | CHEMBL453568)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article