Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50030153
TargetSqualene monooxygenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50032836(4-[(3-{[(6,6-Dimethyl-hept-2-en-4-ynyl)-ethyl-amin...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of pig liver microsomal squalene epoxidase (SE) by measuring the extend of cholesterol radiolabeling after incubation with [14C]m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSqualene monooxygenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291660([3-([3,3']Bithiophenyl-5-ylmethoxy)-benzyl]-ethyl-...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of pig liver microsomal squalene epoxidase (SE) by measuring the extend of cholesterol radiolabeling after incubation with [14C]m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSqualene monooxygenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291661([3-(3-Azido-phenyl)-prop-2-ynyl]-[3-([3,3']bithiop...)
Affinity DataIC50: 270nMAssay Description:In vitro inhibition of pig liver microsomal squalene epoxidase (SE) by measuring the extend of cholesterol radiolabeling after incubation with [14C]m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSqualene monooxygenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291658((3-{[(4-Azido-phenyl)-dimethyl-silanyl]-methoxy}-b...)
Affinity DataIC50: 520nMAssay Description:In vitro inhibition of pig liver microsomal squalene epoxidase (SE) by measuring the extend of cholesterol radiolabeling after incubation with [14C]m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSqualene monooxygenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291659([3-(4-Azido-phenyl)-prop-2-ynyl]-[3-([3,3']bithiop...)
Affinity DataIC50: 960nMAssay Description:In vitro inhibition of pig liver microsomal squalene epoxidase (SE) by measuring the extend of cholesterol radiolabeling after incubation with [14C]m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSqualene monooxygenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291662([3-(2-Azido-phenyl)-prop-2-ynyl]-[3-([3,3']bithiop...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibition of pig liver microsomal squalene epoxidase (SE) by measuring the extend of cholesterol radiolabeling after incubation with [14C]m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article