Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50030100
TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
Affinity DataIC50: 50nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291107((3-Chloro-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-...)
Affinity DataIC50: 100nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291111((6,7-Dimethoxy-quinazolin-4-yl)-methyl-m-tolyl-ami...)
Affinity DataIC50: 180nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291110(Methyl-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)-m-tolyl-...)
Affinity DataIC50: 180nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50273281(CHEMBL456375 | CHEMBL543669 | N-methyl-4-anilino-6...)
Affinity DataIC50: 500nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM6497(6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinazolin...)
Affinity DataIC50: 500nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291103((6,7-Dimethoxy-quinazolin-4-yl)-methyl-(3-trifluor...)
Affinity DataIC50: 500nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM6497(6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinazolin...)
Affinity DataIC50: 500nMAssay Description:Inhibition of p56 lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291112(Methyl-phenyl-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)-a...)
Affinity DataIC50: 600nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291107((3-Chloro-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291109((6,7-Dimethyl-quinazolin-4-yl)-methyl-m-tolyl-amin...)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291116((6,7-Dimethoxy-quinazolin-4-yl)-methyl-p-tolyl-ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291115(Methyl-phenyl-(9H-purin-6-yl)-amine | CHEMBL335052)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291114((4-Chloro-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291114((4-Chloro-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290633(CHEMBL328277 | CHEMBL545776 | 4-(2,3-Dihydro-indol...)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291102((6,7-Dimethoxy-quinazolin-4-yl)-ethyl-phenyl-amine...)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291116((6,7-Dimethoxy-quinazolin-4-yl)-methyl-p-tolyl-ami...)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291115(Methyl-phenyl-(9H-purin-6-yl)-amine | CHEMBL335052)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50273281(CHEMBL456375 | CHEMBL543669 | N-methyl-4-anilino-6...)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291106((2,6-Dichloro-quinazolin-4-yl)-methyl-phenyl-amine...)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50290633(CHEMBL328277 | CHEMBL545776 | 4-(2,3-Dihydro-indol...)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291102((6,7-Dimethoxy-quinazolin-4-yl)-ethyl-phenyl-amine...)
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291109((6,7-Dimethyl-quinazolin-4-yl)-methyl-m-tolyl-amin...)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291111((6,7-Dimethoxy-quinazolin-4-yl)-methyl-m-tolyl-ami...)
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50273281(CHEMBL456375 | CHEMBL543669 | N-methyl-4-anilino-6...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of platelet-derived growth factor receptor (PDGF-R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291104((6-Methoxy-quinazolin-4-yl)-methyl-phenyl-amine; h...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291105((6,8-Dimethyl-quinazolin-4-yl)-methyl-phenyl-amine...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM6497(6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinazolin...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of platelet-derived growth factor receptor (PDGF-R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291104((6-Methoxy-quinazolin-4-yl)-methyl-phenyl-amine; h...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM3260(N-methyl-N-phenylquinazolin-4-amine | 4-Anilino qu...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291101(Methyl-phenyl-(6,7,8-trimethoxy-quinazolin-4-yl)-a...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291101(Methyl-phenyl-(6,7,8-trimethoxy-quinazolin-4-yl)-a...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291105((6,8-Dimethyl-quinazolin-4-yl)-methyl-phenyl-amine...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291106((2,6-Dichloro-quinazolin-4-yl)-methyl-phenyl-amine...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291103((6,7-Dimethoxy-quinazolin-4-yl)-methyl-(3-trifluor...)
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291108((2-Chloro-6,7-dimethoxy-quinazolin-4-yl)-methyl-ph...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291110(Methyl-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)-m-tolyl-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291117(Methyl-phenyl-(2,6,7-trimethoxy-quinazolin-4-yl)-a...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291112(Methyl-phenyl-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)-a...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50291117(Methyl-phenyl-(2,6,7-trimethoxy-quinazolin-4-yl)-a...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM3260(N-methyl-N-phenylquinazolin-4-amine | 4-Anilino qu...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Epidermal growth factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291108((2-Chloro-6,7-dimethoxy-quinazolin-4-yl)-methyl-ph...)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50273281(CHEMBL456375 | CHEMBL543669 | N-methyl-4-anilino-6...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of p56 lck tyrosine kinase (inactive)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM6497(6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinazolin...)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonism towards Colony stimulating factor 1 receptor (CSF-1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article