Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50030003
TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50104969(N-[3-(N'-HYDROXYCARBOXAMIDO)-2-(2-METHYLPROPYL)-PR...)
Affinity DataKi: <10nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50104969(N-[3-(N'-HYDROXYCARBOXAMIDO)-2-(2-METHYLPROPYL)-PR...)
Affinity DataKi: <10nMAssay Description:Inhibition of Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50104969(N-[3-(N'-HYDROXYCARBOXAMIDO)-2-(2-METHYLPROPYL)-PR...)
Affinity DataKi: <10nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50104969(N-[3-(N'-HYDROXYCARBOXAMIDO)-2-(2-METHYLPROPYL)-PR...)
Affinity DataKi: <10nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290164((R)-3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-...)
Affinity DataKi:  184nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290160(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  210nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290163(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  290nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290164((R)-3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-...)
Affinity DataKi:  336nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290160(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  430nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290161(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  550nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290162(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  620nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290162(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  620nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290161(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  640nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290162(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  770nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290164((R)-3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-...)
Affinity DataKi:  860nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290163(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290161(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290161(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290160(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290159(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290160(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290162(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290158(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290158(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  9.90E+3nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290163(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  1.12E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290159(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  1.91E+4nMAssay Description:Inhibition of Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290159(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  1.92E+4nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290158(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi:  2.24E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290164((R)-3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-...)
Affinity DataKi:  2.94E+4nMAssay Description:Inhibition of Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290159(3-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-ethy...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article