Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50029964
TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289733(1-(2,5-Dimethoxy-benzyl)-6-ethoxy-4-(4-methoxy-phe...)
Affinity DataIC50: 200nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289733(1-(2,5-Dimethoxy-benzyl)-6-ethoxy-4-(4-methoxy-phe...)
Affinity DataIC50: 260nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289739(4-Benzo[1,3]dioxol-5-yl-6-ethoxy-1-(2-methoxy-benz...)
Affinity DataIC50: 380nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289739(4-Benzo[1,3]dioxol-5-yl-6-ethoxy-1-(2-methoxy-benz...)
Affinity DataIC50: 450nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289738(6-Ethoxy-1-(2-methoxy-benzyl)-4-(4-methoxy-phenyl)...)
Affinity DataIC50: 500nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289737(4-(2,4-Dimethoxy-phenyl)-6-ethoxy-1-(2-methoxy-ben...)
Affinity DataIC50: 540nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289730(4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 940nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289737(4-(2,4-Dimethoxy-phenyl)-6-ethoxy-1-(2-methoxy-ben...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289732(4-Benzo[1,3]dioxol-5-yl-6-ethyl-1-(2-methoxy-benzy...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289738(6-Ethoxy-1-(2-methoxy-benzyl)-4-(4-methoxy-phenyl)...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289732(4-Benzo[1,3]dioxol-5-yl-6-ethyl-1-(2-methoxy-benzy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289730(4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289734(4-Benzo[1,3]dioxol-5-yl-1-(4-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289731(4-Benzo[1,3]dioxol-5-yl-5,6-dimethoxy-1-(2-methoxy...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289728(4-Benzo[1,3]dioxol-5-yl-1-benzo[1,3]dioxol-5-ylmet...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289728(4-Benzo[1,3]dioxol-5-yl-1-benzo[1,3]dioxol-5-ylmet...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289731(4-Benzo[1,3]dioxol-5-yl-5,6-dimethoxy-1-(2-methoxy...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289734(4-Benzo[1,3]dioxol-5-yl-1-(4-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289736([4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-ox...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289740(4-Benzo[1,3]dioxol-5-yl-1-(3-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289735(4-Benzo[1,3]dioxol-5-yl-1-benzyl-2-oxo-1,2-dihydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289740(4-Benzo[1,3]dioxol-5-yl-1-(3-methoxy-benzyl)-2-oxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289736([4-Benzo[1,3]dioxol-5-yl-1-(2-methoxy-benzyl)-2-ox...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289735(4-Benzo[1,3]dioxol-5-yl-1-benzyl-2-oxo-1,2-dihydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50289729(3-Benzo[1,3]dioxol-5-yl-5-ethoxy-1-(4-methoxy-benz...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of [125I]ET1 binding to rat aorta membranes(ETA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289729(3-Benzo[1,3]dioxol-5-yl-5-ethoxy-1-(4-methoxy-benz...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of [125I]ET1 binding to porcine kidney inner medulla membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article