Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029879
TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288960(N-[(R)-2-(1H-Indol-3-yl)-1-mercaptomethyl-ethyl]-2...)
Affinity DataIC50: 1.70E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288958(2-Biphenyl-4-yl-N-((R)-1-mercaptomethyl-2-pyridin-...)
Affinity DataIC50: 5.20E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288964(Thiophene-2-carboxylic acid [(R)-2-(1H-indol-3-yl)...)
Affinity DataIC50: 5.20E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288957(4-[(R)-2-(1H-Indol-3-yl)-1-mercaptomethyl-ethylcar...)
Affinity DataIC50: 5.40E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288961(1-(2-Biphenyl-4-yl-acetyl)-piperidine-4-carboxylic...)
Affinity DataIC50: 6.50E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288963(2-(4-Benzyloxy-phenyl)-N-[(R)-2-(1H-indol-3-yl)-1-...)
Affinity DataIC50: 6.50E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288962(N-[(R)-2-(1H-Indol-3-yl)-1-mercaptomethyl-ethyl]-2...)
Affinity DataIC50: 7.70E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetEndothelin-converting enzyme 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288959(N-((R)-1-Mercaptomethyl-2-phenyl-ethyl)-nicotinami...)
Affinity DataIC50: 7.80E+3nMAssay Description:Compound was evaluated for inhibition of Endothelin-converting enzyme 1 partially purified from porcine primary aortic endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article