Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50029853
TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataKi:  5nMAssay Description:Inhibition of matrix metalloprotease -1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288702((R)-6-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  8nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288710((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  9.5nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288705((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  10nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288708((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  12nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288704((R)-7-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288716((R)-4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  20nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288707((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  28nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288720((R)-6-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  32nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288716((R)-4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  33nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288717((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  47nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288705((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  60nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288707((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  70nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288715((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  72nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288702((R)-6-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  86nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataKi:  91nMAssay Description:Inhibition of matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288700((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  110nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288708((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  110nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288703((R)-4-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  120nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288711((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  120nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288704((R)-7-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  120nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288715((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  120nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288720((R)-6-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  120nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288713((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  130nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288721((R)-5-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  140nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288701((R)-6-[(1-Acetyl-pyrrolidine-2-carbonyl)-amino]-2-...)
Affinity DataKi:  180nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288709((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  190nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50057083(L-696418 | (R)-2-[(S)-1-(3-Methyl-1-phenylcarbamoy...)
Affinity DataKi:  200nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288718((R)-5-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  270nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288714((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  270nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288712((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  320nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288706((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  350nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288717((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  350nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50057083(L-696418 | (R)-2-[(S)-1-(3-Methyl-1-phenylcarbamoy...)
Affinity DataKi:  470nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288719((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  530nMAssay Description:Inhibition of matrix metalloprotease -3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288721((R)-5-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  570nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288702((R)-6-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  720nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50057083(L-696418 | (R)-2-[(S)-1-(3-Methyl-1-phenylcarbamoy...)
Affinity DataKi:  760nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288714((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  770nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288705((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  870nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288703((R)-4-Benzoylamino-2-[(S)-1-((S)-3-methyl-1-phenyl...)
Affinity DataKi:  1.09E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288712((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288701((R)-6-[(1-Acetyl-pyrrolidine-2-carbonyl)-amino]-2-...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target72 kDa type IV collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288706((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of MMP-2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288708((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288713((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  1.79E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288706((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288716((R)-4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataKi:  2.09E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288710((R)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of matrix metalloprotease -1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Displayed 1 to 50 (of 60 total ) | Next | Last >>
Jump to: