Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50029745
TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287500((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287504((2S,4R)-2-[2-(1,3-Dioxo-1,3-dihydro-benzo[f]isoind...)
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287502(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287502(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287506(4-(1,3-Dioxo-5-propoxy-1,3-dihydro-isoindol-2-yl)-...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287507(4-(5-Methoxy-1,3-dioxo-1,3-dihydro-isoindol-2-yl)-...)
Affinity DataIC50: 570nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287503(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 940nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287503(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 940nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287505(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 970nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287505(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 970nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287497(2-(1-Benzylcarbamoyl-cyclohexylmethyl)-4-(1,3-diox...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287499(4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-{1-[(S)-...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287498(4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl)-2-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287501(2-{1-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbamoyl-e...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against Matrix Metallo Proteinase-1 (MMP-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article