Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50029735
TargetCalpain-1 catalytic subunit(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50073850([(S)-1-(1-Benzyl-2-oxo-ethylcarbamoyl)-2-methyl-pr...)
Affinity DataIC50: 17nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCalpain-1 catalytic subunit(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287391((R)-4-Methyl-2-[2-oxo-2-(9H-xanthen-9-yl)-ethyl]-p...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCalpain-1 catalytic subunit(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287394((R)-2-Isobutyl-4-oxo-5,5-diphenyl-pentanoic acid (...)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCalpain-1 catalytic subunit(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287392((R)-4-Methyl-2-[2-oxo-2-(9H-xanthen-9-yl)-ethyl]-p...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCalpain-1 catalytic subunit(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287390((R)-2-Isobutyl-4-oxo-8-phenyl-octanoic acid ((S)-1...)
Affinity DataIC50: 138nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCalpain-1 catalytic subunit(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287393([(S)-1-(1-Ethylaminooxalyl-propylcarbamoyl)-3-meth...)
Affinity DataIC50: 240nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article