Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50029702
TargetMu-type opioid receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50287045(N-CBM-TAMO | CHEMBL14680)
Affinity DataIC50: 2nMAssay Description:Compound was tested for binding activity against mu opioid receptor in bovine striatal membranes using 0.25 nM [3H]DAMGO as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetD(1A) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50287046(8-Chloro-5-(3-isothiocyanato-phenyl)-3-methyl-2,3,...)
Affinity DataIC50: 2.10nMAssay Description:Compound was tested for binding affinity against Dopamine receptor D1 using 1 nM [3H]SCH-23390 as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287045(N-CBM-TAMO | CHEMBL14680)
Affinity DataIC50: 6.30nMAssay Description:Compound was tested for binding activity against Opioid receptor kappa 1 in bovine striatal membranes using 1 nM [3H]U-69593 as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287045(N-CBM-TAMO | CHEMBL14680)
Affinity DataIC50: 12nMAssay Description:Compound was tested for binding activity against Opioid receptor delta 1 in bovine striatal membranes using 0.2 nM [3H]p-CI-DPDPE as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50287046(8-Chloro-5-(3-isothiocyanato-phenyl)-3-methyl-2,3,...)
Affinity DataIC50: 978nMAssay Description:Compound was tested for binding affinity against Dopamine receptor D2 using 10 nM [3H]N-methyl-spiperone as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article