Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50029641
LigandPNGBDBM50286446({(S)-1-[(S)-1-(4-Hydroxy-benzyl)-2-oxo-ethylcarbam...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286452({(S)-1-[(S)-1-(4-Hydroxy-benzyl)-2-oxo-ethylcarbam...)
Affinity DataIC50: 25nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286449({(S)-1-[(S)-1-(4-Methoxy-benzyl)-2-oxo-ethylcarbam...)
Affinity DataIC50: 30nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50137397([(S)-1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-3-methy...)
Affinity DataIC50: 35nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50014577(CHEMBL286722 | benzyl (S)-3-methyl-1-oxo-1-((S)-1-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50073850([(S)-1-(1-Benzyl-2-oxo-ethylcarbamoyl)-2-methyl-pr...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286453({(S)-1-[(S)-1-(4-Hydroxy-benzyl)-2-oxo-ethylcarbam...)
Affinity DataIC50: 55nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286455([(S)-1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-3,3-dim...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286454([(S)-1-((S)-1-Formyl-2-naphthalen-1-yl-ethylcarbam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286445([((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-phenyl-methyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286444([(S)-1-((S)-1-Formyl-3-phenyl-propylcarbamoyl)-2-m...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286443([(S)-1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-ethyl]-...)
Affinity DataIC50: 140nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286456([(S)-1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-3-pheny...)
Affinity DataIC50: 270nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286450([(S)-1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-2-pheny...)
Affinity DataIC50: 400nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286451([1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-2,2-dimethy...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286448([(S)-1-((S)-1-Benzyl-2-oxo-ethylcarbamoyl)-2-napht...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50286447([1-(2-Formyl-pyrrolidine-1-carbonyl)-2-methyl-prop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Calpain 1 by [3H]acetyl-casein assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article