Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50029416
TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284287(Endothelin-1 analogue | CHEMBL438213)
Affinity DataIC50: 7.53E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284290(Endothelin-1 analogue | CHEMBL412233)
Affinity DataIC50: 9.93E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284275(Endothelin-1 analogue | CHEMBL414596)
Affinity DataIC50: 8.06E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284289(Endothelin-1 analogue | CHEMBL382683)
Affinity DataIC50: 7.60E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284282(Endothelin-1 analogue | CHEMBL411290)
Affinity DataIC50: 1.00E+7nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284285(Endothelin-1 analogue | CHEMBL440254)
Affinity DataIC50: 6.85E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284286(Endothelin-1 analogue | CHEMBL411371)
Affinity DataIC50: 8.60E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284277(Endothelin-1 analogue | CHEMBL411933)
Affinity DataIC50: 9.40E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284288(Endothelin-1 analogue | CHEMBL439090)
Affinity DataIC50: 5.77E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284290(Endothelin-1 analogue | CHEMBL412233)
Affinity DataIC50: 1.01E+7nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284289(Endothelin-1 analogue | CHEMBL382683)
Affinity DataIC50: 1.00E+7nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284283(Endothelin-1 analogue | CHEMBL439489)
Affinity DataIC50: 8.89E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284279(Endothelin-1 analogue | CHEMBL439471)
Affinity DataIC50: 7.97E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284287(Endothelin-1 analogue | CHEMBL438213)
Affinity DataIC50: 9.40E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284288(Endothelin-1 analogue | CHEMBL439090)
Affinity DataIC50: 7.96E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284278(Endothelin-1 analogue | CHEMBL383109)
Affinity DataIC50: 7.55E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284275(Endothelin-1 analogue | CHEMBL414596)
Affinity DataIC50: 9.78E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284281(Endothelin-1 analogue | CHEMBL383113)
Affinity DataIC50: 7.04E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284284(Endothelin-1 analogue | CHEMBL216868)
Affinity DataIC50: 6.71E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284280(Endothelin-1 analogue | CHEMBL411360)
Affinity DataIC50: 9.05E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284286(Endothelin-1 analogue | CHEMBL411371)
Affinity DataIC50: 6.07E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284285(Endothelin-1 analogue | CHEMBL440254)
Affinity DataIC50: 8.60E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284284(Endothelin-1 analogue | CHEMBL216868)
Affinity DataIC50: 9.77E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284283(Endothelin-1 analogue | CHEMBL439489)
Affinity DataIC50: 9.76E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284282(Endothelin-1 analogue | CHEMBL411290)
Affinity DataIC50: 9.88E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284281(Endothelin-1 analogue | CHEMBL383113)
Affinity DataIC50: 9.59E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284280(Endothelin-1 analogue | CHEMBL411360)
Affinity DataIC50: 9.00E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284279(Endothelin-1 analogue | CHEMBL439471)
Affinity DataIC50: 9.94E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284278(Endothelin-1 analogue | CHEMBL383109)
Affinity DataIC50: 6.13E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284276(Endothelin-1 analogue | CHEMBL264220)
Affinity DataIC50: 5.27E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284277(Endothelin-1 analogue | CHEMBL411933)
Affinity DataIC50: 7.59E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET A receptor obtained from rat thoracic aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284276(Endothelin-1 analogue | CHEMBL264220)
Affinity DataIC50: 5.59E+6nMAssay Description:Concentration required to produce 50% inhibition of binding against ET B receptor obtained from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article