Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50029372
TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283886(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283895(3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-1,7...)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283891(2-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283899(ethyl[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-o...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283888(4-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283892(3-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283901(Staurosporine derivative | CHEMBL335931)
Affinity DataIC50: 160nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283894(3-methoxy-2-methyl-4-methylamino-(2R,3S,4S,6S)-29-...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283892(3-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283909(1N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa...)
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283900(4-ethyl(methyl)amino-3-methoxy-2-methyl-(2R,3S,4S,...)
Affinity DataIC50: 240nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283903(18-hydroxy-5-methoxy-6-methyl-4-methylamino-(2S,4S...)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283900(4-ethyl(methyl)amino-3-methoxy-2-methyl-(2R,3S,4S,...)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 350nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283886(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50: 600nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283894(3-methoxy-2-methyl-4-methylamino-(2R,3S,4S,6S)-29-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM31094(PKC-412 | cid_24202429)
Affinity DataIC50: 800nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283902(4-benzyl(methyl)amino-3-methoxy-2-methyl-(2R,3S,4S...)
Affinity DataIC50: 910nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283896(N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283906(2-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283883(methyl 2-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283887(4-[2-hydroxyhexyl(methyl)amino]-3-methoxy-2-methyl...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283903(18-hydroxy-5-methoxy-6-methyl-4-methylamino-(2S,4S...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31094(PKC-412 | cid_24202429)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283889(Staurosporine derivative | CHEMBL130049)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283893(1N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283901(Staurosporine derivative | CHEMBL335931)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283882(3-methoxy-4-[4-methoxyphenyl(methyl)carboxamido]-2...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283898(4-[3-chlorophenyl(methyl)carboxamido]-3-methoxy-2-...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283897(4-[2-chlorophenyl(methyl)carboxamido]-3-methoxy-2-...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283904(3-methoxy-2-methyl-4-methyl(3-nitrophenyl)carboxam...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283912(1N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283910(4-[4-chlorophenyl(methyl)carboxamido]-3-methoxy-2-...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283878(Staurosporine derivative | CHEMBL336192)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283905(3-methoxy-2-methyl-4-methyl(2-pyrazinyl)carboxamid...)
Affinity DataIC50: 8.18E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283881(3-methoxy-2-methyl-4-methyl(3-pyridyl)carboxamido-...)
Affinity DataIC50: 8.18E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283879(3-methoxy-2-methyl-4-methyl[methylamino(thioxo)met...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283884(Staurosporine derivative | CHEMBL338449)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283880(4-[3,5-dinitrophenyl(methyl)carboxamido]-3-methoxy...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283911(methyl 2-[3-methoxy-2-methyl-4-methyl(phenyl)carbo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283914(17-benzyl-3-methoxy-2-methyl-4-methyl(phenyl)carbo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article