Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029278
TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50093095(2-[(S)-1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)...)
Affinity DataIC50: 0.530nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50154572(2-[1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2,2...)
Affinity DataIC50: 0.850nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281976(2-Benzhydryl-3-(3,5-dimethyl-benzyloxy)-1-aza-bicy...)
Affinity DataIC50: 1nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282931(2-[1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-e...)
Affinity DataIC50: 2.20nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282923([(R)-1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl...)
Affinity DataIC50: 4.40nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282925([(S)-1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl...)
Affinity DataIC50: 5.5nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282927([1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-eth...)
Affinity DataIC50: 6.80nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50154580(1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-ethy...)
Affinity DataIC50: 9.30nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282933(1-(3-Bromo-5-methyl-benzyloxymethyl)-2,2-diphenyl-...)
Affinity DataIC50: 9.70nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50154571(1-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-2,2-di...)
Affinity DataIC50: 10.7nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282935(N-[1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-e...)
Affinity DataIC50: 11nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282929(1-(3,5-Dichloro-benzyloxymethyl)-2,2-diphenyl-ethy...)
Affinity DataIC50: 11.3nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282932([1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-eth...)
Affinity DataIC50: 12.7nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282938(1-(3,5-Dibromo-benzyloxymethyl)-2,2-diphenyl-ethyl...)
Affinity DataIC50: 13.3nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282923([(R)-1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl...)
Affinity DataIC50: 14nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282926(3-(3,5-Dimethyl-benzyloxy)-1,1-diphenyl-propan-2-o...)
Affinity DataIC50: 17nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282936(N-[1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-e...)
Affinity DataIC50: 21nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282928([1-(3,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-eth...)
Affinity DataIC50: 55nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282924(1-(3-Chloro-benzyloxymethyl)-2,2-diphenyl-ethylami...)
Affinity DataIC50: 75nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282937(1-(3-Iodo-benzyloxymethyl)-2,2-diphenyl-ethylamine...)
Affinity DataIC50: 77nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282930(Benzyl-[1-(3,5-dimethyl-benzyloxymethyl)-2,2-diphe...)
Affinity DataIC50: 82nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282922(Cyclopropylmethyl-[1-(3,5-dimethyl-benzyloxymethyl...)
Affinity DataIC50: 93nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282934(1-(2,5-Dimethyl-benzyloxymethyl)-2,2-diphenyl-ethy...)
Affinity DataIC50: 150nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSubstance-P receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50154573(1-Benzyloxymethyl-2,2-diphenyl-ethylamine | CHEMBL...)
Affinity DataIC50: 367nMAssay Description:Binding affinity towards human Tachykinin receptor 1 expressed in CHO cells by the displacement of [125 I] substance PMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article