Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50029109
TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281565((S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045240(Ac-D-Phe-Leu-Phe-Ile-Ile-Trp | (S)-2-[(S)-2-((2S,5...)
Affinity DataIC50: 35nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281564((S)-4-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: 650nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045227(Ac-D-Phe-Orn-Asp-Ile-Ile-Trp | (S)-3-[2-((R)-2-Ace...)
Affinity DataIC50: 750nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281565((S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)
Affinity DataIC50: 930nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045240(Ac-D-Phe-Leu-Phe-Ile-Ile-Trp | (S)-2-[(S)-2-((2S,5...)
Affinity DataIC50: 1.18E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281564((S)-4-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045227(Ac-D-Phe-Orn-Asp-Ile-Ile-Trp | (S)-3-[2-((R)-2-Ace...)
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045258((S)-2-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)
Affinity DataIC50: 8.00E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045251(Ac-D-Phe-Asp-Ile-Ile-Trp | 3-((R)-2-Acetylamino-3-...)
Affinity DataIC50: 9.10E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045251(Ac-D-Phe-Asp-Ile-Ile-Trp | 3-((R)-2-Acetylamino-3-...)
Affinity DataIC50: 9.30E+3nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50000566((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 9.50E+3nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045235((S)-3-[(R)-2-((1S,5S)-2-Acetylamino-3-phenyl-propi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000566((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045235((S)-3-[(R)-2-((1S,5S)-2-Acetylamino-3-phenyl-propi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045258((S)-2-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045247(Ac-D-Phe-Ile-Ile-Trp | 3-((R)-2-Acetylamino-3-phen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045247(Ac-D-Phe-Ile-Ile-Trp | 3-((R)-2-Acetylamino-3-phen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045248((S)-3-[(S)-2-((S)-2-Acetylamino-3-phenyl-propionyl...)
Affinity DataIC50: 1.84E+4nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50045248((S)-3-[(S)-2-((S)-2-Acetylamino-3-phenyl-propionyl...)
Affinity DataIC50: 1.85E+4nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [125I]ET1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article