Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50029051
TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50280989(2,6-dimethyl-5-methyloxycarbonyl-4-(3-nitrophenyl)...)
Affinity DataIC50: 16nMAssay Description:Tested for its inhibitory activity against Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280989(2,6-dimethyl-5-methyloxycarbonyl-4-(3-nitrophenyl)...)
Affinity DataIC50: 295nMAssay Description:Tested for its ability to inhibit the binding of [125I]ET1 to the Endothelin B receptor in rat cerebellum membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50280990(2,6-dimethyl-5-methyloxycarbonyl-4-(3-nitrophenyl)...)
Affinity DataIC50: 422nMAssay Description:Tested for its inhibitory activity against Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280989(2,6-dimethyl-5-methyloxycarbonyl-4-(3-nitrophenyl)...)
Affinity DataIC50: 592nMAssay Description:Inhibition of [3H]PN-200-110 binding to L-type calcium channels in rat cortex membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280990(2,6-dimethyl-5-methyloxycarbonyl-4-(3-nitrophenyl)...)
Affinity DataIC50: 2.70E+3nMAssay Description:Tested for its inhibitory activity against Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article