Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50029025
LigandPNGBDBM50001266(CHEMBL50267 | 5,7-dichlorokynurenic acid | 5,7-Dic...)
Affinity DataKi:  40nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50004952(CHEMBL31344 | 3-(2-Carboxy-ethyl)-4,6-dichloro-1H-...)
Affinity DataKi:  140nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50129080(3-Carboxymethyl-4,6-dichloro-1H-indole-2-carboxyli...)
Affinity DataKi:  340nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280807(3-Carboxymethyl-5,7-dichloro-4-oxo-1,4-dihydro-qui...)
Affinity DataKi:  650nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50004960(CHEMBL301556 | 4,6-Dichloro-1H-indole-2-carboxylic...)
Affinity DataKi:  980nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50009092(CHEMBL23754 | 3-Carboxymethyl-1H-indole-2-carboxyl...)
Affinity DataKi:  5.24E+3nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM81975(4-hydroxyquinoline-2-carboxylic acid | NSC_5280455...)
Affinity DataKi:  5.40E+3nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280805(3-(2-Carboxy-ethyl)-5,7-dichloro-4-oxo-1,4-dihydro...)
Affinity DataKi:  7.04E+3nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280806(3-Carboxymethyl-4-oxo-1,4-dihydro-quinoline-2-carb...)
Affinity DataKi:  1.48E+4nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50009085(CHEMBL25599 | 3-Carboxymethyl-quinoline-2-carboxyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Tested for the ability to displace [3H]glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article