Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50028942
LigandPNGBDBM50280269(3-[2-(4-Amino-benzylcarbamoyl)-ethyl]-4,6-dichloro...)
Affinity DataIC50: 27nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50061396(4,6-Dichloro-3-(2-phenylcarbamoyl-ethyl)-1H-indole...)
Affinity DataIC50: 36nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50004952(CHEMBL31344 | 3-(2-Carboxy-ethyl)-4,6-dichloro-1H-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280277(3-Carbamoyl-6-chloro-1H-indole-2-carboxylic acid |...)
Affinity DataIC50: 810nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50009079(CHEMBL415462 | 6-Chloro-3-methoxycarbonylmethyl-1H...)
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280272(6-Chloro-3-hydroxymethyl-1H-indole-2-carboxylic ac...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280270((2R,3R)-3-Carbamoyl-6-chloro-2,3-dihydro-1H-indole...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280273((2R,3R)-3-Benzoyloxymethyl-6-chloro-2,3-dihydro-1H...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280274((2R,3R)-6-Chloro-2,3-dihydro-1H-indole-2,3-dicarbo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280275((2R,3R)-6-Chloro-3-hydroxymethyl-2,3-dihydro-1H-in...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280276((2R,3R)-3-Carboxymethyl-6-chloro-2,3-dihydro-1H-in...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280278((R)-6-Chloro-1,2-dihydro-indole-2,3,3-tricarboxyli...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280271((2R,3R)-6-Chloro-2,3-dihydro-1H-indole-2,3-dicarbo...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of [3H]L-689,560 binding to Glycine site of NMDA receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article