Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50023628
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of PI3Kdelta (unknown origin) preincubated for 30 mins followed by ATP addition and measured after 1 hrs by ADP-Glo reagent based analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 589nMAssay Description:Inhibition of PI3Kalpha (unknown origin) preincubated for 30 mins followed by ATP addition and measured after 1 hrs by ADP-Glo reagent based analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 605nMAssay Description:Inhibition of PI3Kgamma (unknown origin) preincubated for 30 mins followed by ATP addition and measured after 1 hrs by ADP-Glo reagent based analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) preincubated for 30 mins followed by ATP addition and measured after 1 hrs by ADP-Glo reagent based analysisMore data for this Ligand-Target Pair
