Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50035561
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026279(3-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026297(4-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026288(3-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026298(3-{2-[2-(2-tert-Butoxycarbonylamino-acetylamino)-3...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026299(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026286(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026284(2-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026283(1-(2-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026282(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026291(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026295(3-{2-[2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-p...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026296(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367238(CHEMBL1790763)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026290(3-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026292(2-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026280(2-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026293(3-({1-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026281(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026294([1-[1-(1-Carbamoyl-ethylcarbamoyl)-3-methyl-butylc...)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50144035((S)-2-(4-Chloro-benzoylamino)-3-(1H-indol-3-yl)-pr...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026285(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50014888(CHEMBL316561 | 4-Benzoylamino-4-dipropylcarbamoyl-...)
Affinity DataIC50: 2.50E+6nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026287(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed