Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50022170
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Affinity DataKd:  188nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 0.140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 0.420nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648947(CHEMBL5613749)
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 5.10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648948(CHEMBL5613986)
Affinity DataIC50: 9.30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648952(CHEMBL5612816)
Affinity DataIC50: 23nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648952(CHEMBL5612816)
Affinity DataIC50: 31nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 31nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 32nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648952(CHEMBL5612816)
Affinity DataIC50: 42nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648949(CHEMBL5612781)
Affinity DataIC50: 49nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM440444(US10633389, Example 109-3 | US20230279020, Example...)
Affinity DataIC50: 73nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 138nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50609301(CHEMBL4559961)
Affinity DataIC50: 181nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtein arginine N-methyltransferase 3(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 321nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 321nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648952(CHEMBL5612816)
Affinity DataIC50: 343nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 351nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 555nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 1.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 1.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 2.40E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 5.90E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 7.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 8.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Affinity DataIC50: 1.00E+6nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Affinity DataIC50: 1.00E+7nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Affinity DataIC50: 1.00E+7nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50648946(CHEMBL5613649)
Affinity DataIC50: 1.00E+7nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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