Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50022233
Affinity DataEC50: 12nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 410nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 560nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.86E+3nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+3nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >3.10E+3nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+3nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 4.30E+3nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+3nMAssay Description:Induction of N-terminal HiBiT tag knocked in IKZF3 degradation in human DF15 cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of C-terminal HiBiT tag knocked in SALL4 degradation in human NCCIT cells incubated for 60 mins by Nano-Glo HiBiT lytic reagent based assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged CK1alpha degradation in human MDS-L cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair
TargetEukaryotic peptide chain release factor GTP-binding subunit ERF3A(Human)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of ePL tagged GSPT1 degradation in human DF15 cells incubated for 60 mins by luminescence reader assayMore data for this Ligand-Target Pair


















