Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 5759
TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93124(Trisubsituted thiazole, 14)
Affinity DataIC50: 6.60E+3nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93125(Trisubsituted thiazole, 15)
Affinity DataIC50: 1.25E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93130(Trisubsituted thiazole, 29)
Affinity DataIC50: 1.25E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93129(Trisubsituted thiazole, 23)
Affinity DataIC50: 1.53E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93124(Trisubsituted thiazole, 14)
Affinity DataIC50: 2.94E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93127(Trisubsituted thiazole, 17)
Affinity DataIC50: 3.30E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93128(Trisubsituted thiazole, 20)
Affinity DataIC50: 3.30E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93131(Trisubsituted thiazole, 30)
Affinity DataIC50: 3.30E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 2a(malaria parasite P. falciparum)
University, Mississippi

LigandPNGBDBM93126(Trisubsituted thiazole, 16)
Affinity DataIC50: 3.91E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93125(Trisubsituted thiazole, 15)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93126(Trisubsituted thiazole, 16)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93127(Trisubsituted thiazole, 17)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93128(Trisubsituted thiazole, 20)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93130(Trisubsituted thiazole, 29)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93131(Trisubsituted thiazole, 30)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article

TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
University, Mississippi

LigandPNGBDBM93129(Trisubsituted thiazole, 23)
Affinity DataIC50: 5.52E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2013
Entry Details Article