Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50020806
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633714(CHEMBL5413186)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of human PD-L1/PD-L1 interaction incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633708(CHEMBL5413429)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of PD-L1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM575481(US11459339, Example 1 | N,N′-(2,2′-dim...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human PD-L1/PD-L1 interaction incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633707(CHEMBL5398154)
Affinity DataIC50: 0.480nMAssay Description:Inhibition of PD-L1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50629797(CHEMBL5403219)
Affinity DataIC50: 0.930nMAssay Description:Inhibition of PD-1/PD-L1 (unknown origin) protein-protein interactionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM491037(US10975049, Example 4 | (S) N-(4-(2-bromo-3-phenyl...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50239948(US9850225, Example 1166 | CHEMBL4071326)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633716(CHEMBL5427239)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human PD-1/PD-L1 interaction overexpressed in human HEK293T cells by flow cytometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633717(CHEMBL5397229)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PD-1/PD-L1 interaction (unknown origin) by AlphaLISA assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50578293(CHEMBL4873960)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PD-1/PD-L1 interaction (unknown origin) by AlphaLISA assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM395411((R)-1-((7-cyano-2-(3′-(3-(((R)-3-hydroxypyrr...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human PD-L1/PD-L1 interaction incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633713(CHEMBL5420708)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of PD-1/PD-L1 (unknown origin) interactionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633712(CHEMBL5416779)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of PD-1/PD-L1 (unknown origin) interaction incubated for 2 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633715(CHEMBL5431974)
Affinity DataIC50: 18nMAssay Description:Inhibition of human PD-1/PD-L1 interaction incubated for 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Henan University

Curated by ChEMBL
LigandPNGBDBM50239947(US9872852, Example 202 | CHEMBL4089730 | US2023030...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human PD-L1 (18 to 134 residues) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr by spectrophometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Henan University

Curated by ChEMBL
LigandPNGBDBM50405449(CHEMBL5266711)
Affinity DataIC50: 22nMAssay Description:Inhibition of human PD-L1 expressed in Escherichia coli BL21 (DE3) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633709(CHEMBL5399462)
Affinity DataIC50: 23nMAssay Description:Inhibition of PD-1/PD-L1 interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50587736(PYRVINIUM | CHEBI:8687 | Pyrvinium | Pyrvinium (ca...)
Affinity DataIC50: 30nMAssay Description:Inhibition of PD-1/PD-L1 (unknown origin) protein-protein interaction incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Henan University

Curated by ChEMBL
LigandPNGBDBM50405450(CHEMBL5315609)
Affinity DataIC50: 43nMAssay Description:Inhibition of human PD-L1 expressed in Escherichia coli BL21 (DE3) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM491038(US10975049, Example 6 | (S)-isopropyl N-(4-(2-brom...)
Affinity DataIC50: 45nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633711(CHEMBL5430522)
Affinity DataIC50: 57nMAssay Description:Inhibition of PD-1/PD-L1 (unknown origin) interaction incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Henan University

Curated by ChEMBL
LigandPNGBDBM50239943(US9872852, Example 8 | CHEMBL4099869)
Affinity DataIC50: 146nMAssay Description:Inhibition of human PD-L1 (18 to 134 residues) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr by spectrophometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50585850(CHEMBL5087003)
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of human PD-1/PD-L1 interaction incubated for 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM50633710(CHEMBL5401124)
Affinity DataIC50: 8.52E+3nMAssay Description:Inhibition of PD-1/PD-L1 (unknown origin) interaction incubated for 15 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Henan University

Curated by ChEMBL
LigandPNGBDBM643925(US11866416, Compound SN-I-240j)
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of human PD-1/PD-L1 interaction incubated for 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed